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GSK-3β inhibitor 14
CAS No. 863004-48-2
GSK-3β inhibitor 14( —— )
Catalog No. M36031 CAS No. 863004-48-2
GSK-3β inhibitor 14 (1,5-Benzothiazepin-4(5H)-one, 2,3-dihydro-2-methyl-5-(phenylmethyl)-) is a weak GSK-3β inhibitor, IC50﹥ 100μM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 134 | In Stock |
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| 5MG | 198 | In Stock |
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| 10MG | 301 | In Stock |
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| 25MG | 466 | In Stock |
|
| 50MG | 624 | In Stock |
|
| 100MG | 826 | In Stock |
|
| 200MG | 1098 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameGSK-3β inhibitor 14
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NoteResearch use only, not for human use.
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Brief DescriptionGSK-3β inhibitor 14 (1,5-Benzothiazepin-4(5H)-one, 2,3-dihydro-2-methyl-5-(phenylmethyl)-) is a weak GSK-3β inhibitor, IC50﹥ 100μM.
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DescriptionGSK-3β inhibitor 14 (Compound 6i), benzothiazepinone derivative, is a weak GSK-3β inhibitor (IC50 >100 μM).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayPI3K/Akt/mTOR signaling
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TargetGSK-3
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RecptorGSK-3
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Research Area——
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Indication——
Chemical Information
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CAS Number863004-48-2
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Formula Weight283.39
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Molecular FormulaC17H17NOS
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Purity>98% (HPLC)
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Solubility——
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SMILESC(N1C=2C(SC(C)CC1=O)=CC=CC2)C3=CC=CC=C3
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Zhang P, et al. Design, synthesis and biological evaluation of benzothiazepinones (BTZs) as novel non-ATP competitive inhibitors of glycogen synthase kinase-3β (GSK-3β). Eur J Med Chem. 2013 Mar;61:95-103.?
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